Nootropique Modafinil

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Tout le modafinil naturel a la stГ©rГ©ochimie R. Modafinil est le nom chimique du composГ© N-Г©thylamphГ©tamine. On pense que le modafinil libГЁre de l'acГ©tyl-Г©thylcholine (AEC), l'un des nombreux agonistes des rГ©cepteurs nicotiniques de l'acГ©tylcholine, dans le cerveau. Il est fabriquГ© sous forme de poudre cristalline blanche Г  blanc cassГ©. Le modafinil et ses mГ©tabolites ont une affinitГ© de liaison trГЁs Г©levГ©e pour le cytochrome P450, en particulier le CYP2C9.

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Le modafinil ne traverse pas la barriГЁre hГ©mato-encГ©phalique. Une dose unique de modafinil dure gГ©nГ©ralement de 6 Г  8 heures. Les principaux mГ©tabolites du modafinil sont le desmГ©thylcitalopram et le N-desmГ©thylmodafinil. Les effets secondaires peuvent inclure des maux de tГЄte, des troubles du sommeil et des nausГ©es. Le modafinil n'amГ©liore pas l'Г©veil pendant la journГ©e, seulement la nuit.
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